ChiiArtesunate?
Artesunate mushonga unorwisa marariya. Iyo inonyungudika nemvura hemisuccinate kubva kune dihydroartemisinin.
Artemisinin is a sesquiterpene lactone yakaparadzaniswa neArtemisia annua, muriwo wagara uchishandiswa kuChina kurapa marariya.
Artesunateuye metabolite yayo inoshanda dihydroartemisinin ine simba reropa schizonticides, inoshanda padanho rering yeparasite. Artesunate yakanakira kurapa marariya yakanyanya, kusanganisira cerebral malaria. Inoshanda zvakare kurwisa chloroquine uye mefloquine isingagadzirirwe mhando dzeP. falciparum. Iyo haina kugadzikana mune isina kwayakarerekera mhinduro uye saka inowanikwa chete kune majekiseni se artesunic acid. Majekiseni anogadzirwa anofanira kugadzirirwa pakarepo asati ashandiswa mu5% (w/v) sodium bicarbonate solution kugadzira munyu sodium artesunate.
Zita | Artesunate |
CAS NO. | 88495-63-0 |
Molecular formula | C19H28O8 |
Assay | 99% |
Hunhu | White crystalline powder |
Molecular uremu | 384.42 |
1.Artesunate ine basa rekudzora vivax marariya uye falciparum marariya chiratidzo, pamwe nekurapa kwechloroquine-resistant rudzi rwezvipembenene.
2. Artesunate ine basa reoxidant. artemisinin inoderedzwa ne catalase, dithiothreitol uye alpha tocopherol.
3.Artesunate nebasa reantibacterial, artemisinin ine anti-influenza virus effect.
4.Artesunate nebasa re-anti-parasite, artemisinin pane basa re-anti-schistosomiasis uye leptospirosis.
ONGORORO | KUTAURA | RESULTS |
Chitarisiko | Bvisa hupfu chena | Zvinoenderana |
Kunhuwa | Hunhu | Zvinoenderana |
tsanangudzo | Nobiletin 98% | Zvinoenderana |
Sieve analysis | 100% inopfuura 80 mesh | Zvinoenderana |
Kurasika paKuomesa | ≤5.0% | Zvinoenderana |
Residue paIgnition | ≤5.0% | Zvinoenderana |
Heavy Metal | Zvinoenderana | |
As | ≤1ppm | Zvinoenderana |
Residual Solvents | EP2000 | Zvinoenderana |
Residual Pesticide | Negative | Zvinoenderana |
Microbiology | ||
Total Plate Count | Zvinoenderana | |
Yeast & Mold | Zvinoenderana | |
E.Coli | Negative | Zvinoenderana |
Salmonella | Negative | Zvinoenderana |
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